Inhibitors

Loline
Catalog No: CFN00291

Loline can reduce prolactin release at the highest concentration, 10(-4) M.

Laurifoline
Catalog No: CFN97205

Laurifoline is a potential NF-κB inhibitor and a potential β2 -adrenegic receptor agonist, it can not only inhibit Pseudomonas aeruginosa PAK strain-induced inflammatory responses via a negative regulation of the Braf protein that participates in MAPK signaling pathway but also activate the β2 -adrenegic receptor. Laurifoline may show anti-HBV activities in vitro using the HBV transfected Hep G2.2.15 cell line.

27-p-Coumaroyloxyursolic acid
Catalog No: CFN97217

27-trans-p-Coumaroyloxyursolic acid and 27-cis-p-coumaroyloxyursolic acid show potent inhibitory activity in the acyl CoA cholesteryl acyl transferase (ACAT) assay.

Acetylursolic acid
Catalog No: CFN97219

Acetylursolic acid shows significant cytotoxic activities, and shows suppression of the SOS-inducing activity of mutagenic heterocyclic amine, Trp-P-1. 3β-Acetylursolic acid can reduce parasitaemia against Plasmodium berghei.

8-Geranyloxypsoralen
Catalog No: CFN97225

8-Geranyloxypsoralen inhibits β-secretase (BACE1) activity in non-competitive manner, with the IC(50) values <25.0 uM, it can induce vasorelaxation on rat arterial tissues. 8-Geranyloxypsoralen possesses nematicidal activities, the median lethal concentrations (LC(50)) is 188.3 mg/ L against B. xylophilus and is 117.5 mg/L against P. redivivus.